XIMELAGATRAN

XIMELAGATRAN

Stock Code: 3575358
Manufacturer Part No: SML1768-25MG
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£806.46 (exc VAT) per 25MG
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Biochem/physiol Actions


Ximelagatran is orally active, selective and potent direct thrombin inhibitor. Ximelagatran is a prodrug of thrombin inhibitor melagatran.


It inhibits both clot-bound and free thrombin. It is quickly absorbed by the small intestine and converted to its active dipeptide drug form, Melagatran. Melagatran associates with the arginine side pocket in thrombin and inactivates it. Ximelagatran has a half-life of 4-5 hours. It is administered orally twice a day.


Packaging


5, 25 mg in glass bottle

Colourwhite to beige
Quality Level100
InChI keyZXIBCJHYVWYIKI-PZJWPPBQSA-N
InChI1S/C24H35N5O5/c1-2-34-20(30)15-26-21(17-6-4-3-5-7-17)24(32)29-13-12-19(29)23(31)27-14-16-8-10-18(11-9-16)22(25)28-33/h8-11,17,19,21,26,33H,2-7,12-15H2,1H3,(H2,
ManufacturerSIGMA-ALDRICH
SolubilityDMSO: 20 mg/mL, clear
Formpowder
Assay≥98% (HPLC)

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