MLS1547

MLS1547

Stock Code: 3574758
Manufacturer Part No: SML1331-25MG
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£391.39 (exc VAT) per 25MG
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Biochem/physiol Actions


MLS1547 is a highly efficacious D2 dopamine receptor (D2R) G protein-biased agonist that does not recruit β-arrestin, and is an antagonist of dopamine-stimulated β-arrestin recruitment to the D2 receptor. MLS-1547 is the first D2 receptor agonist with close to full efficacy for G protein signaling (EC50 = 370 nM), but no ability to recruit β-arrestin.


Packaging


5, 25 mg in glass bottle

Colourwhite to beige
Quality Level100
InChI keyOPEJNANYABTIGC-UHFFFAOYSA-N
InChI1S/C19H19ClN4O/c20-16-12-14(19(25)18-15(16)4-3-7-22-18)13-23-8-10-24(11-9-23)17-5-1-2-6-21-17/h1-7,12,25H,8-11,13H2
ManufacturerSIGMA-ALDRICH
SolubilityDMSO: 5 mg/mL, clear (warmed)
Formpowder
Assay≥98% (HPLC)

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