BIM5078

BIM5078

Stock Code: 3574098
Manufacturer Part No: SML0528-25MG
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£619.82 (exc VAT) per 25MG
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Biochem/physiol Actions


BIM5078 is a potent Hepatocyte nuclear factor 4a (HNF4a) antagonist that directly binds to ligand-binding pocket and modulates the expression of known HNF4a target genes. BIM5078 also inhibits insulin gene expression by disruption of E47 and PDX-1 binding to insulin promoter. BIM5078 is selectively cytotoxic to transformed cells.


Features and Benefits


This compound is a featured product for Gene Regulation research. Click here to discover more featured Gene Regulation products. Learn more about bioactive small molecules for other areas of research at sigma.com/discover-bsm.


Packaging


5, 25 mg in glass bottle

Colourwhite to beige
Quality Level100
InChI keyDLUVMRPVZILBOE-UHFFFAOYSA-N
InChI1S/C14H10ClN3O4S/c1-9-16-12-4-2-3-5-13(12)17(9)23(21,22)14-8-10(18(19)20)6-7-11(14)15/h2-8H,1H3
ManufacturerSIGMA-ALDRICH
SolubilityDMSO: 10 mg/mL, clear (warmed)
Formpowder
Assay≥98% (HPLC)

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