ASP7663

ASP7663

Stock Code: 3574950
Manufacturer Part No: SML1467-25MG
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£667.18 (exc VAT) per 25MG
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Biochem/physiol Actions


ASP7663 is a selective activator of transient receptor potential ankyrin 1 (TRPA1), known to play a role for chemical sensing in the pain pathway. ASP7663 activated human, rat, and mouse TRPA1 receptors with EC50 values of 510, 540, and 500 nM, respectively, and little or no affinity at more than 60 other related receptors, channels and enzymes. ASP7663 enhanced colonic motility and exerted analgesic effects against abdominal pain in mouse models.


Packaging


5, 25 mg in glass bottle

Colourlight orange to dark orange
Quality Level100
InChI keyRCVZUIGCNAAMIC-UXBLZVDNSA-N
InChI1S/C14H14FNO3/c1-8(2)7-16-13-9(4-3-5-11(13)15)10(14(16)19)6-12(17)18/h3-6,8H,7H2,1-2H3,(H,17,18)/b10-6+
ManufacturerSIGMA-ALDRICH
SolubilityDMSO: 25 mg/mL, clear
Formpowder
Assay≥98% (HPLC)

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