GSK137647A

GSK137647A

Biochem/physiol Actions

GSK137647A is a selective agonist of the free fatty acid receptor 4 (FFA4/GPR120), which is involved in long-chain fatty acid stimulated GLP-1 secretion and has been implicated in glucose homeostasis, adiposity, and regulation of the anti-inflammatory response. GSK137647A has pEC50 values of 6.3, 6.2, and 6.1 for human, mouse and rat FFA4, and pEC50 values ﹤ 4.5 for all three species for FFA1, FFA2, and FFA3.

Packaging

5, 25 mg in glass bottle

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Code Description Colour Quality Level InChI key InChI Manufacturer Solubility Form Assay Price Quantity
3574534 GSK137647A white to beige 100 FQUAFMNPXPXOJE-UHFFFAOYSA-N 1S/C16H19NO3S/c1-11-9-12(2)16(13(3)10-11)17-21(18,19)15-7-5-14(20-4)6-8-15/h5-10,17H,1-4H3
£551.57 (exc VAT) per 25MG
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3574535 GSK137647A white to beige 100 FQUAFMNPXPXOJE-UHFFFAOYSA-N 1S/C16H19NO3S/c1-11-9-12(2)16(13(3)10-11)17-21(18,19)15-7-5-14(20-4)6-8-15/h5-10,17H,1-4H3
£136.50 (exc VAT) per 5MG
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