CRT0066101 HYDROCHLORIDE

Biochem/physiol Actions

CRT0066101 is a very potent inhibitor of Protein Kinase D (PKD) isoforms with IC50 values for PKD-1, -2 and -3 = 1, 2.5 and 2 nM, respecitively. CRT0066101 has been shown to have anticancer activity. CRT0066101 potently inhibits proliferation of PANC-1 pancreatic cells, and blocks migration and invasion of U87MG glioblastoma cells. CRT0066101 has also been shown to decrease growth of primary tumors and metastasis of ER(-) breast cancers.

Packaging

5 mg in glass bottle

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Code Description Colour Quality Level Manufacturer Storage Temp. Solubility Form Assay Price Quantity
3575002 CRT0066101 HYDROCHLORIDE white to beige 100 SIGMA-ALDRICH −20°C
£502.82 (exc VAT) per 25MG
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3575003 CRT0066101 HYDROCHLORIDE white to beige 100 SIGMA-ALDRICH −20°C
£135.80 (exc VAT) per 5MG
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