BX-912

BX-912

Biochem/physiol Actions

BX-912 is a potent inhibitor of PDK1 (3-Phosphoinositide dependent protein kinase-1). The IC50 values for direct inhibition of kinase activity or inhibition in a cell based assay are 26 nM and 12 nM, respectively. BX-912 inhibits the growth of PC-3 tumor cells grown on soft agar more potently than cells grown on plastic (IC50 = 320 nM vs. 5.5 mM, respectively).

Packaging

5, 25 mg in glass bottle

No detailed specifications are available for this product.

There are no downloads for this product.

Code Description Colour Quality Level Manufacturer Storage Temp. Solubility Form Assay Price Quantity
3574450 BX-912 white to beige 100 SIGMA-ALDRICH −20°C DMSO: 10 mg/mL, clear powder ≥95% (HPLC)
£357.96 (exc VAT) per 25MG
-
+
3574451 BX-912 white to beige 100 SIGMA-ALDRICH −20°C DMSO: 10 mg/mL, clear powder ≥95% (HPLC)
£122.43 (exc VAT) per 5MG
-
+